{"id":319933,"date":"2022-03-24T09:34:37","date_gmt":"2022-03-24T09:34:37","guid":{"rendered":"https:\/\/afrikmag.com\/var\/www\/vhosts\/afrikmag.compublic_html\/?p=319933"},"modified":"2022-03-24T09:34:53","modified_gmt":"2022-03-24T09:34:53","slug":"une-pilule-contraceptive-pour-homme-efficace-a-99-sur-les-souris","status":"publish","type":"post","link":"https:\/\/afrikmag.com\/var\/www\/vhosts\/afrikmag.compublic_html\/une-pilule-contraceptive-pour-homme-efficace-a-99-sur-les-souris\/","title":{"rendered":"Une pilule contraceptive pour homme efficace \u00e0 99 % sur les souris"},"content":{"rendered":"\n<p class=\"wp-block-paragraph\">Les scientifiques travaillant sur une pilule contraceptive pour homme ont d\u00e9couvert que le m\u00e9dicament \u00e9tait efficace \u00e0 99% pour pr\u00e9venir la grossesse chez la souris.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">La nouvelle pilule contraceptive pour homme non hormonale qui perturbe une prot\u00e9ine particuli\u00e8re impliqu\u00e9e dans la formation des spermatozo\u00efdes, a montr\u00e9 une pr\u00e9vention efficace de la grossesse, une r\u00e9versibilit\u00e9 en quelques semaines et aucun effet secondaire observable.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Les chercheurs de l&rsquo;Universit\u00e9 du Minnesota ont pr\u00e9sent\u00e9 les r\u00e9sultats de leur essai mercredi 23 mars, lors de la r\u00e9union de printemps de l&rsquo;American Chemical Society (ACS).&nbsp;&nbsp;\u00c0 l&rsquo;heure actuelle, il n&rsquo;existe que deux options de contraception efficaces pour les hommes; les pr\u00e9servatifs et la vasectomie.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">La nouvelle pilule contraceptive masculine cible une prot\u00e9ine appel\u00e9e RAR-\u03b1 (RAR-alpha). Cette prot\u00e9ine joue un r\u00f4le, entre autres, dans la diff\u00e9renciation cellulaire, qui comprend la production de sp3rme. Des \u00e9tudes ant\u00e9rieures ont montr\u00e9 que faire taire le g\u00e8ne RAR-\u03b1 chez les souris les rend st\u00e9riles.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Gunda Georg, chef du d\u00e9partement de chimie m\u00e9dicinale de l&rsquo;universit\u00e9, a d\u00e9clar\u00e9 que les tests de la pilule, YCT529, qui s&rsquo;est av\u00e9r\u00e9e \u00abefficace \u00e0 99% chez la souris\u00bb, seront utilis\u00e9s dans des essais cliniques humains qui commenceront au troisi\u00e8me ou quatri\u00e8me trimestre de&nbsp;&nbsp;2022.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Georg a dit: \u00ab&nbsp;<em>Parce qu&rsquo;il peut \u00eatre difficile de pr\u00e9dire si un compos\u00e9 qui semble bon dans les \u00e9tudes sur les animaux se d\u00e9roulera \u00e9galement dans les essais sur l&rsquo;homme, nous explorons actuellement d&rsquo;autres compos\u00e9s \u00e9galement\u00a0\u00bb.<\/em><\/p>\n\n\n\n<p class=\"wp-block-paragraph\">L&rsquo;ACS a \u00e9galement d\u00e9clar\u00e9 que la pilule, qui limite les chances de f\u00e9condation des femelles, perd son effet lorsqu&rsquo;elle n&rsquo;est plus prise.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">La d\u00e9claration se lit comme suit: \u00ab<em>Pour d\u00e9velopper leur contraceptif masculin non hormonal, les chercheurs ont cibl\u00e9 une prot\u00e9ine appel\u00e9e r\u00e9cepteur alpha de l&rsquo;acide r\u00e9tino\u00efque (RAR-\u03b1). Cette prot\u00e9ine fait partie d&rsquo;une famille de trois r\u00e9cepteurs nucl\u00e9aires qui se lient \u00e0 l&rsquo;acide r\u00e9tino\u00efque, une forme de vitamine A qui joue un r\u00f4le important dans la croissance cellulaire, la diff\u00e9renciation (y compris la formation des spermatozo\u00efdes) et le d\u00e9veloppement embryonnaire. L&rsquo;inactivation du g\u00e8ne RAR-\u03b1 chez les souris m\u00e2les les rend st\u00e9riles, sans aucun effet secondaire \u00e9vident.<\/em>&nbsp;<em>D&rsquo;autres scientifiques ont d\u00e9velopp\u00e9 un compos\u00e9 oral qui inhibe les trois membres de la famille RAR (RAR-\u03b1, -\u03b2 et -\u03b3) et provoque une st\u00e9rilit\u00e9 r\u00e9versible chez les souris m\u00e2les, mais l&rsquo;\u00e9quipe de Georg et leurs collaborateurs en biologie de la reproduction voulaient trouver un m\u00e9dicament qui \u00e9tait&nbsp;&nbsp;sp\u00e9cifiques pour RAR-\u03b1 et donc moins susceptibles de provoquer des effets secondaires.<\/em><\/p>\n\n\n\n<p class=\"wp-block-paragraph\">LIRE AUSSI: <a href=\"https:\/\/afrikmag.com\/var\/www\/vhosts\/afrikmag.compublic_html\/sante-une-pilule-contraceptive-masculine-sans-hormones-en-cours-de-developpement\/\">Sant\u00e9: Une pilule contraceptive masculine en cours de d\u00e9veloppement<\/a><\/p>\n\n\n\n<p class=\"wp-block-paragraph\"><em>Les chercheurs ont donc examin\u00e9 de pr\u00e8s les structures cristallines des RAR-\u03b1, -\u03b2 et -\u03b3 li\u00e9s \u00e0 l&rsquo;acide r\u00e9tino\u00efque, identifiant les diff\u00e9rences structurelles dans la mani\u00e8re dont les trois r\u00e9cepteurs se lient \u00e0 leur ligand commun. Avec ces informations, ils ont con\u00e7u et synth\u00e9tis\u00e9 environ 100 compos\u00e9s et \u00e9valu\u00e9 leur capacit\u00e9 \u00e0 inhiber s\u00e9lectivement RAR-\u03b1 dans les cellules. Ils ont identifi\u00e9 un compos\u00e9, nomm\u00e9 YCT529, qui inhibait RAR-\u03b1 presque 500 fois plus puissamment que RAR-\u03b2 et -\u03b3. Lorsqu&rsquo;il a \u00e9t\u00e9 administr\u00e9 par voie orale \u00e0 des souris m\u00e2les pendant 4 semaines, YCT529 a consid\u00e9rablement r\u00e9duit le nombre de spermatozo\u00efdes et a \u00e9t\u00e9 efficace \u00e0 99% pour pr\u00e9venir la grossesse, sans aucun effet secondaire observable.&nbsp;&nbsp;Les souris pouvaient \u00e0 nouveau engendrer des petits 4 \u00e0 6 semaines apr\u00e8s avoir cess\u00e9 de recevoir le compos\u00e9.\u00bb<\/em><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Les scientifiques travaillant sur une pilule contraceptive pour homme ont d\u00e9couvert que le m\u00e9dicament \u00e9tait efficace \u00e0 99% pour pr\u00e9venir la grossesse chez la souris. La nouvelle pilule contraceptive pour homme non hormonale qui perturbe une prot\u00e9ine particuli\u00e8re impliqu\u00e9e dans la formation des spermatozo\u00efdes, a montr\u00e9 une pr\u00e9vention efficace de la grossesse, une r\u00e9versibilit\u00e9 en &hellip;<\/p>\n","protected":false},"author":37,"featured_media":319952,"comment_status":"open","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[371,7020],"tags":[14732,1403,10857,7901],"class_list":["post-319933","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-sante","category-societe","tag-contraceptifs","tag-hommes","tag-pilule","tag-souris"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v28.5 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Une pilule contraceptive pour homme efficace \u00e0 99 % sur les souris<\/title>\n<meta name=\"description\" content=\"Les scientifiques travaillant 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